Consecutive Reactions with Sulfoximines: Straightforward Synthesis of Substituted 5,5-Spiroketals
نویسندگان
چکیده
منابع مشابه
Synthesis and bioactivity of new phosphorylated R,R'-substituted sulfoximines.
R,R'-disubstituted sulfoximines were phosphorylated with O,O-diethylchloro phosphate and phosphorothionate to obtain new organophosphorus compounds. After purification they were characterized by GC-MS and (1)H-NMR. The toxicity of the synthesized O,O-diethyl N-(R,R'-disubstituted sulfoximine) phosphoro-amidothionates was assayed on Musca domestica. It was found that the methyl phenyl derivative...
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Spiroketals are widely found as substructures of many naturally occurring compounds from diverse sources including plants, animals as well as microbes. Naturally occurring spiroketals are biologically active and most of them are chiral molecules. This article aims at reviewing the asymmetric synthesis of biologically active spiroketals for last 10 years (1998-2007).
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ژورنال
عنوان ژورنال: Synthesis
سال: 2011
ISSN: 0039-7881,1437-210X
DOI: 10.1055/s-0030-1260039